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Solid-phase organik syntheses - Burdges K.

Burdges K. Solid-phase organik syntheses - John Wiley & Sons, 2000. - 283 p.
ISBN 0-471-22824-9
Download (direct link): phaseorganicsynthesis2000.pdf
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58. Sarges, R.; Lyga, J. W. Synthesis and Aldose Reductase Inhibitory Activity of N-l,N-4-Disubstituted 3,4-Dihydro-2(lH)-quinoxalinone Derivatives, J. Heterocycl. Chem. 1988, 25, 1475.
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27, 50. Mebendazole and Related Antihelmintics, Van den Bossche, H.; Rochette, F.; Hoerig, C. Adv. Pharmacol. Chemother. 1982, 79, 67.
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61. Phillips, G. B.; Wei, G. P. Solid Phase Synthesis of Benzimidazoles, Tetrahedron Lett. 1996, 37, 4887.
62. Kugishima, H.; Horie, ̉.; Imafuku, K. Synthesis of 3-[[(2-Benzimida-zolyl)thio]methyl]-1 -methyl-1,8-dihydrocycloheptapyrazol-8-ones, J. Het-erocycl. Chem. 1994, 31, 1557.
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64. Saluja, S.; Zou, R.; Drach, J. C.; Townsend, L. B. Structure-Activity Relationships among 2-Substituted 5,6-Dichloro-, 4,6-Dichloro- and 4,5-Di-chloro-1-[(2-hydroxyethoxy)methyl]- and -1-[(1,3-dihydroxy-2-propoxy)methyl]benzimidazoles, J. Med. Chem. 1996, 39, 881.
65. Ellingboe, J. W.; Spinelli, W.; Winkley, M. W.; Nguyen, ̉. ̉.; Parsons, R. W.; Moubarak, I. F.; Kitzen, J. ̀.; Von Engen, D.; Bagli, J. F. Class III Antiarrhythmic Activity of Novel Substituted 4-[(Methylsulfonyl)amino]-benzamides and Sulfonamides, J. Med. Chem. 1992, 35, 705.
66. Holmes, D. S.; Bethell, R. C.; Cammack, N.; Clemens, I. R.; Kitchin, J.; McMeekin, P.; Mo, C. L.; Orr, D. C.; Patel, B. et al. Synthesis and Structure-Activity Relationships of a Series of Penicillin-derived HIV Proteinase Inhibitors Containing a Stereochemically Unique Peptide Isostere, J. Med. Chem. 1993, 36, 3129.
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68. Schwarz, ̀. K.; Gallop, M. A., unpublished results.
69. Studies on the Chemistry of Thienoannulated 0,N- and S,N-Containing Heterocycles. 1. Nucleophilic Substitution Reactions on Chlorinated Thio-phene Derivatives as a Basis for the Synthesis of Thienoannulated 0,N- and
S,N-Heterocycles, Puschmann, I.; Erker, T. Heterocycles 1993,36,1323. See also: Studies on the Chemistry of Thienoanellated 0,N- and S,N-Containing Heterocycles. II. Synthesis on Thieno-Dilthiazem Analogs, Puschmann, I.; Erker, T. Heterocycles 1995, 41, 709.
Solid-Phase Organic Synthesis. Edited by Kevin Burgess Copyright © 2000 John Wiley & Sons, Inc. ISBNs: 0-471-31825-6 (Hardback); 0-471-22824-9 (Electronic)
(iv) repeat
JEFFREY S. MOORE, DAVID J. HILL, and MATTHEW J. MIO The University of Illinois at Urbana-Champaign
Solid-phase organic synthesis (SPOS) is an established technique for generation of peptides,1,2 nucleotides,3 and more recently, carbohydrates (oligosaccharides).4-5 Supported syntheses of nonbiological oligomers6-16 and other small molecules17-21 have also been reported, reflecting the method’s
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