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Solid-phase organik syntheses - Burdges K.

Burdges K. Solid-phase organik syntheses - John Wiley & Sons, 2000. - 283 p.
ISBN 0-471-22824-9
Download (direct link): phaseorganicsynthesis2000.pdf
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Jiong Chen, Texas A & M University, Department of Chemistry, PO Box 30012, College Station, TX 77842-3012, USA
Rajesh V. Devraj, Parallel Medicinal & Combinatorial Chemistry Unit, Searle/Monsanto Life Sciences Company, 800 N. Lindbergh Blvd., St. Louis, MO 63167, USA
Nicholas J. Ede, Chiron Technologies Pty. Ltd., 11 Duerdin St., Clayton, Victoria, 3168 Australia
Mark A. Gallop, Affymax Research Institute, 4001 Miranda Avenue, Palo Alto, CA 94304, USA email: Mark_Gallop@affymax.com
xiv CONTRIBUTORS
Daniel L. Flynn, Amgen, One Amgen Center Drive, Thousand Oaks, CA 91320-1799, USA email: dflynn@amgen.com
David J. Hill, The University of Illinois at Urbana-Champaign, Roger Adams Laboratory, Box 55-5, 600 South Mathews, Urbana, IL 61801, USA
Ian W. James, Chiron Technologies Pty. Ltd., 11 Duerdin St., Clayton, Victoria, 3168 Australia email: Ian_James@cc.chiron.com
Matthew J. Mio, The University of Illinois at Urbana-Champaign, Roger Adams Laboratory, Box 55-5, 600 South Mathews, Urbana, IL 61801, USA
Jeffrey S. Moore, The University of Illinois at Urbana-Champaign, Roger Adams Laboratory, Box 55-5, 600 South Mathews, Urbana, IL 61801, USA
email: moore@aries.scs.uiuc.edu
John J. Parlow, Parallel Medicinal & Combinatorial Chemistry Unit, Searle/Monsanto Life Sciences Company, 800 N. Lindbergh Blvd., St. Louis, MO 63167, USA
Matthias K. Schwarz, Serono Pharmaceutical Research Institute, 14 che-min des Aulx, CH-1228 Plan-les-Ouates, Geneva, Switzerland email: Matthias .Schwarz @ serono.com
Matthew H. Todd, Department of Chemistry, University of California, Berkeley, CA 94720, USA
Geoffrey Wickham, Chiron Technologies Pty. Ltd., 11 Duerdin St., Clayton, Victoria, 3168 Australia
Lawrence J. Wilson, Proctor & Gamble Pharmaceuticals, 8700 Mason-Montgomery Road, Mason, OH 45040, USA email: wilsonlj@pg.com
Bing Yan, Novartis Pharmaceuticals Corporation. 556 Morris Avenue, Summit, NJ 07901, USA email: bin.yan@pharma.Novartis.com
SOLID-PHASE ORGANIC SYNTHESIS
Agitation, effects on reaction rates,
237 Aldehydes, 88
Aldose reductase inhibitors, 100 Alkene metathesis, 253 Alkylation reactions, 8 allylic, palladium catalyzed, 69, 169 N-, 42, 93, 97 reductive, 34 S-, 106 Alkylboranes, 50 Alkynes, silylated, 32, 38 Allyl carbonate, 69 Allyl silane, 60
Amine oxides as cooxidants, 168 Amino acids, 100 bicyclic, 41 N-methyl, 101 spirocyclic, 101 P-, 92, 93 (5-, esters of, 95 Aminoiminomethanesulfonic acid, 6 Aminomethyl polystyrene, 18, 152,
165
Aminophosphorane, 8 Aminothiazoles, 157, 160 Angiotensin receptor antagonists, 68 Anilines, 30, 84, 86, 88, 93, 101, 102, 105, 107, 260 halo-, 34 iodo-, 32, 33 Anthranilic acids, 93 Antiarrhymic agents, 107 Antisense oligonucleotides, 16 Antiviral agents, 107 Aperiodic sequences of oligomers, 120 ArgoGel resin, 58 Armstrong, 52, 54, 55 Attenuated total reflectance, 222, 223 Aza-Wittig, 8, 9, 206 Azodicarboxylates, 161
Baccatin, 256 Balanol, 261 BBN, 9-, 60,61,62 Beam condensers, 222
270 INDEX
Benzaldehydes, 86 Benzamide, 4-fluoro-3-nitro, 97 Benzimidates, 105, 106 Benzimidazoles, 105 Benzimidazolones, 84, 106 aminomethyl-, 84 thio-, 84 Benzodiazepines, 47, 102, 200 2,5-diones, 50 receptor, partial agonists, 99 Benzodiazepinones, 93, 95, 96 Benzofuran, 30, 35 Benzoic acids 4-fluoro-3-nitro, 82, 84, 102, 104 iodo-, 45, 50 Benzothiazapinones, 84 Benzothiazepine, 92 Benzothiazepines, 84, 109 Benzothiazepinones, 88, 91, 92, 109 Benzothiazocinones, 84, 89, 92 Benzotriazoles, 87, 88 Biaryls, 25, 45, 49, 55, 59, 63 Biguanide, 10 Biphenyls, 45 Birefringence, 136 Bisborylation reactions, 52 Bishydroxylations, 171 Boronates, 48, 55 pinacol, 50, 54 vinyl, 53, 54 Boronic acids, 48, 49, 50, 51, 57, 67 Brandykinin antagonist, 68 Bromination, 182 Bromoketones, 157 Burgessí reagent, 7, 166
Calcium antagonists, 84 * Carbamates, supported, 164 Carbamimidothioates, methyl, 4
Carbodiimides, 6, 7, 8, 9, 93, 206 DCC, 126 DIC, 45, 88 EDC, 11, 14, 20, 160 supported form of EDC, 186 Carbomoylguanidines, 11 Carbonate, allyl, 69 Carbon-carbon bond formation, 25, 172
Carbonimidates, diphenyl, 3 Carboxyimidazole, 11 Cardiovascular disorders, 84 Catalysis, rates on solid phases, 238 Catalysts, immobilized, 26 Cesium carbonate, 49 Chlorination, 3
Chloromethyl polystyrene, 39, 253, 255
oxidation of, 254 Cholecystokinin A receptor, 200 Chromates, polymer-supported, 168 Cinchona alkaloid, polymer-supported for bishydroxylations, 171 Cleavage. See Resin cleavage Cobalt catalysis, 170 Complementary molecular reactivity sequestrants, 152 Compression cell, 222 Condensation reactions, 160 Condensations, ketophosphonate-aldehyde, 255 Convergent syntheses of dendrimers, 133
Copper catalysis, 48 Copper(l+) iodide, 30 Corey-Kim oxidations, 255 COSY, 138
Cross-site reactivity, 152 Crowns. See Pins Cuprates, 248, 251, 255 Cyanamides, 4 Cyanogen bromide, 4
INDEX 271
Cyclin-dependent kinases, 202 Cyclization, 38. See macrocyclization Cycloadditions [2+2], 57 1,3-dipolar, 263 Cyclooxygenase, 66 Cyclotryprostatins, 260 Cysteine, 92, 109
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